Protease Inhibitors and Phosphatase Inhibitors
MilliporeSigma™ Calbiochem™ Apoptosis Inhibitor
The Apoptosis Inhibitor, also referenced under CAS 54135-60-3, controls the biological activity of Apoptosis. This small molecule/inhibitor is primarily used for Cancer applications.
MilliporeSigma™ Calbiochem™ Apocynin
A cell-permeable, anti-inflammatory phenolic compound that acts as a potent and selective inhibitor of NADPH oxidase.
MilliporeSigma™ Calbiochem™ Bax-Inhibiting Peptide, V5
A cell-permeable pentapeptide based on the Ku70-Bax inhibiting domain that offers cytoprotection.
MilliporeSigma™ Calbiochem™ MCT1 Inhibitor, SR13800
A cell-permeable inhibitor of monocarboxylate transporter 1 (MCT1). Blocks the proliferation of Raji Burkitt lymphoma cells expressing MCT1 (EC50 = 5 nM).
MilliporeSigma™ Calbiochem™ InSolution™ Akt Inhibitor X
The InSolution™ Akt Inhibitor X, also referenced under CAS 925681-41-0, controls the biological activity of Akt. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
MilliporeSigma™ Calbiochem™ Akt Inhibitor X
The Akt Inhibitor X, also referenced under CAS 925681-41-0, controls the biological activity of Akt. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
MilliporeSigma™ Calbiochem™ β-Glucuronidase Inhibitor
The β-Glucuronidase Inhibitor controls the biological activity of β-Glucuronidase.
MilliporeSigma™ Calbiochem™ Ghrelin Receptor Antagonist, JMV 2959
A 1, 2, 4-triazole derived compound that acts as a potent ghrelin receptor (GHS-R1a) antagonist (IC50 = 32nM in a binding assay, dissociation constant Kb =
MilliporeSigma™ Calbiochem™ ISR Inhibitor, ISRIB
The cell-permeable, selective inhibitor of eIF2α/eIF2S1 Ser51 phosphorylation-initiated UPR response (≈25 to 200 nM) upon ER stress induction.
MilliporeSigma™ Calbiochem™ Sodium Orthovanadate, Activated
A depolymerized vanadate prepared from Sodium Orthovanadate with enhanced ability to competitively inhibit endogenous phosphatases.
MP Biomedicals™ Protease Inhibitor Cocktail Kit
Research Use Only
MilliporeSigma™ Calbiochem™ Phosphatase Inhibitor Cocktail Set III
Phosphatase Inhibitor Cocktail Set III is a ready to use cocktail of four phosphatase inhibitors for broad-spectrum inhibition of both serine/threonine and protein tyrosine phosphatases.
MilliporeSigma™ Calbiochem™ Phenylmethylsulfonyl Fluoride
Phenylmethylsulfonyl Fluoride, CAS 329-98-6, is an irreversible inhibitor of serine proteases. It causes sulfonylation of the active-site serine residues.
MilliporeSigma™ Calbiochem™ PPACK, Dihydrochloride
PPACK, Dihydrochloride, CAS 142036-63-3, is an extremely potent and selective irreversible inhibitor of thrombin (Kobs/[I] = 107M-1S-1). Reacts with thrombin in a 1:1 stoichiometry.
MilliporeSigma™ Calbiochem™ PP1 Analog II, 1NM-PP1
PP1 Analog II, CAS 221244-14-0, is a cell-permeable PP1 analog that acts as a potent, reversible, selective, ATP-competitive inhibitor of mutant over wild-type kinases.